High Potency VEGFRs/MET/FMS Triple Blockade by TAS-115 Concomitantly Suppresses Tumor Progression and Bone Destruction in Tumor-Induced Bone Disease Model with Lung Carcinoma Cells.
第一作者:
Hidenori,Fujita
第一单位:
Discovery and Preclinical Research Division, Taiho Pharmaceutical Co., Ltd., Tsukuba, Ibaraki, Japan.
作者:
主题词
动物(Animals);骨肿瘤(Bone Neoplasms);细胞分化(Cell Differentiation);细胞增殖(Cell Proliferation);疾病模型, 动物(Disease Models, Animal);人类(Humans);吲哚类(Indoles);肺肿瘤(Lung Neoplasms);男(雄)性(Male);小鼠(Mice);小鼠, 近交BALB C(Mice, Inbred BALB C);小鼠, 裸(Mice, Nude);破骨细胞(Osteoclasts);蛋白激酶抑制剂(Protein Kinase Inhibitors);原癌基因蛋白质c-met(Proto-Oncogene Proteins c-met);吡唑类(Pyrazoles);吡啶类(Pyridines);吡咯类(Pyrroles);喹啉类(Quinolines);RANK配体(RANK Ligand);受体, 巨噬细胞集落刺激因子(Receptor, Macrophage Colony-Stimulating Factor);受体, 血管内皮生长因子(Receptors, Vascular Endothelial Growth Factor);信号传导(Signal Transduction);硫脲(Thiourea);胫骨(Tibia);移植, 异种(Transplantation, Heterologous);X线显微体层摄影术(X-Ray Microtomography)
DOI
10.1371/journal.pone.0164830
PMID
27736957
发布时间
2018-12-11
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PloS one
e0164830页
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