Caffeic acid phenethyl ester (CAPE) revisited: Covalent modulation of XPO1/CRM1 activities and implication for its mechanism of action.
作者:
主题词
结合部位(Binding Sites);咖啡酸类(Caffeic Acids);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);人类(Humans);核胞浆转运蛋白类(Karyopherins);质谱分析法(Mass Spectrometry);显微镜检查, 共焦(Microscopy, Confocal);分子动力学模拟(Molecular Dynamics Simulation);肽类(Peptides);苯乙基醇(Phenylethyl Alcohol);蛋白质结构, 三级(Protein Structure, Tertiary);受体, 胞质和核(Receptors, Cytoplasmic and Nuclear);构效关系(Structure-Activity Relationship)
DOI
10.1111/cbdd.12905
PMID
27863053
发布时间
2023-12-13
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Chemical biology & drug design
655-662页
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