A fluorescence-based high-throughput assay to identify inhibitors of tyrosylprotein sulfotransferase activity.
第一作者:
Wenbo,Zhou
第一单位:
Center for Drug Design, Academic Health Center, University of Minnesota, 516 Delaware St. SE, 7-215 PWB, MMC 204, Minneapolis, MN 55455, USA.
作者:
主题词
杆状病毒科(Baculoviridae);色谱法, 液相(Chromatography, Liquid);组合化学技术(Combinatorial Chemistry Techniques);剂量效应关系, 药物(Dose-Response Relationship, Drug);荧光(Fluorescence);人类(Humans);半数抑制浓度(Inhibitory Concentration 50);同工酶类(Isoenzymes);动力学(Kinetics);肽类(Peptides);底物特异性(Substrate Specificity);磺基转移酶类(Sulfotransferases);舒拉明(Suramin);串联质谱法(Tandem Mass Spectrometry)
DOI
10.1016/j.bbrc.2016.12.013
PMID
27923653
发布时间
2018-01-18
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