From Homology Models to a Set of Predictive Binding Pockets-a 5-HT<sub>1A</sub> Receptor Case Study.
第一作者:
Dawid,Warszycki
第一单位:
Institute of Pharmacology, Polish Academy of Sciences , 12 Smetna Street, 31-343 Kraków, Poland.
作者:
医学主题词
结晶学, X线(Crystallography, X-Ray);药物评价, 临床前(Drug Evaluation, Preclinical);HEK293细胞(HEK293 Cells);人类(Humans);配体(Ligands);蒙特卡罗法(Monte Carlo Method);蛋白质结合(Protein Binding);蛋白质构象(Protein Conformation);受体, 血清素, 5-HT1A(Receptor, Serotonin, 5-HT1A);结构同源性, 蛋白质(Structural Homology, Protein)
DOI
10.1021/acs.jcim.6b00263
PMID
28055203
发布时间
2023-11-04
基金项目
R01 GM071872/GM/NIGMS NIH HHS/United States
R01 GM074832/GM/NIGMS NIH HHS/United States
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