RXRα ligand Z-10 induces PML-RARα cleavage and APL cell apoptosis through disrupting PML-RARα/RXRα complex in a cAMP-independent manner.
第一作者:
Lin,Xu
第一单位:
School of Pharmaceutical Sciences, Fujian Provincial Key Laboratory of Innovative Drug Target Research, Xiamen University, Xiamen, Fujian, China.
作者:
主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);砷剂(Arsenicals);印迹法, 蛋白质(Blotting, Western);COS细胞(COS Cells);半胱氨酸天冬氨酸蛋白酶(Caspases);细胞系, 肿瘤(Cell Line, Tumor);环AMP(Cyclic AMP);流式细胞术(Flow Cytometry);HEK293细胞(HEK293 Cells);人类(Humans);白血病, 早幼粒细胞, 急性(Leukemia, Promyelocytic, Acute);配体(Ligands);萘类(Naphthalenes);硝基化合物(Nitro Compounds);癌基因蛋白质类, 融合(Oncogene Proteins, Fusion);氧化物(Oxides);蛋白质结合(Protein Binding);维甲类X受体α(Retinoid X Receptor alpha);苯乙烯类(Styrenes);维甲酸(Tretinoin)
DOI
10.18632/oncotarget.14812
PMID
28129653
发布时间
2019-12-10
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Oncotarget
12311-12322页
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