Identification of novel dual-specificity phosphatase 26 inhibitors by a hybrid virtual screening approach based on pharmacophore and molecular docking.
第一作者:
Ji-Xia,Ren
第一单位:
Institute of Medicinal Plant Development, Chinese Academy of Medical Science & Peking Union Medical College, 151 Malianwa North Road, Haidian District, Beijing 100193, China,; College of Life Science, Liaocheng University, Liaocheng 252059, Shandong, China.
作者:
主题词
氨基酸序列(Amino Acid Sequence);结合部位(Binding Sites);计算机模拟(Computer Simulation);药物评价, 临床前(Drug Evaluation, Preclinical);双特异性磷酸酶类(Dual-Specificity Phosphatases);酶抑制剂(Enzyme Inhibitors);丝裂原活化蛋白激酶磷酸酶类(Mitogen-Activated Protein Kinase Phosphatases);模型, 化学(Models, Chemical);模型, 分子(Models, Molecular);蛋白质构象(Protein Conformation)
DOI
10.1016/j.biopha.2017.02.064
PMID
28249240
发布时间
2018-02-20
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