Epidermal growth factor receptor (EGFR) structure-based bioactive pharmacophore models for identifying next-generation inhibitors against clinically relevant EGFR mutations.
第一作者:
Pooja S,Panicker
第一单位:
Centre for Nanosciences and Molecular Medicine, Amrita Institute of Medical Sciences and Research Centre, Amrita University, Kochi, Kerala, India.
作者:
主题词
抗肿瘤药(Antineoplastic Agents);计算机辅助设计(Computer-Aided Design);药物设计(Drug Design);人类(Humans);羟肟酸类(Hydroxamic Acids);突变(Mutation);蛋白激酶抑制剂(Protein Kinase Inhibitors);量化构效关系(Quantitative Structure-Activity Relationship);喹唑啉类(Quinazolines);小分子化合物库(Small Molecule Libraries)
DOI
10.1111/cbdd.12977
PMID
28303669
发布时间
2018-12-02
- 浏览60

Chemical biology & drug design
629-636页
相似文献
- 中文期刊
- 外文期刊
- 学位论文
- 会议论文