Topical Intestinal Aminoimidazole Agonists of G-Protein-Coupled Bile Acid Receptor 1 Promote Glucagon Like Peptide-1 Secretion and Improve Glucose Tolerance.
作者:
主题词
胺化作用(Amination);动物(Animals);Caco-2细胞(Caco-2 Cells);糖尿病, 2型(Diabetes Mellitus, Type 2);胰高血糖素样肽1(Glucagon-Like Peptide 1);葡萄糖(Glucose);葡糖耐量试验(Glucose Tolerance Test);人类(Humans);降血糖药(Hypoglycemic Agents);咪唑类(Imidazoles);肠吸收(Intestinal Absorption);肠黏膜(Intestinal Mucosa);小鼠, 近交C57BL(Mice, Inbred C57BL);受体, G-蛋白偶联(Receptors, G-Protein-Coupled)
DOI
10.1021/acs.jmedchem.6b01873
PMID
28414465
发布时间
2018-12-30
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Journal of medicinal chemistry
4185-4211页
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