Synthesis of 3- and 29-substituted celastrol derivatives and structure-activity relationship studies of their cytotoxic activities.
第一作者:
Wei-Guang,Shan
第一单位:
College of Pharmaceutical Science, Zhejiang University of Technology, Hangzhou 310014, PR China.
作者:
主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞系, 肿瘤(Cell Line, Tumor);细胞存活(Cell Survival);药物设计(Drug Design);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);酯化(Esterification);人类(Humans);小鼠, 裸(Mice, Nude);肿瘤(Neoplasms);五环三萜类(Pentacyclic Triterpenes);构效关系(Structure-Activity Relationship);三萜类(Triterpenes)
DOI
10.1016/j.bmcl.2017.05.083
PMID
28587825
发布时间
2021-12-04
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