Inhibition of the endocannabinoid-regulating enzyme monoacylglycerol lipase elicits a CB<sub>1</sub> receptor-mediated discriminative stimulus in mice.
第一作者:
Robert A,Owens
第一单位:
Department of Pharmacology and Toxicology, Medical College of Virginia Campus, Virginia Commonwealth University, Richmond, VA, USA.
作者:
关键词
2-Arachidonoylglycerol (2-AG)Alpha/beta-hydrolase domain 6 (ABHD6)CP55,940 (PubChem CID: 104895)Cannabinoid-1 (CB1) receptorDiazepam (PubChem CID: 3016)Discriminative stimulusDrug discriminationEndogenous cannabinoidsFatty acid amide hydrolase (FAAH)JZL184 (PubChem CID: 25021165)KT182 (PubChem CID: 53364491)MJN110 (PubChem CID: 71722059)Monoacylglycerol lipase (MAGL)N-arachidonoylethanolamine (anandamide,?AEA)Nicotine (PubChem CID: 24278591)PF-3845 (PubChem CID: 25154867)Rimonabant (PubChem CID: 104850)SA-57 (PubChem CID: 44589122)Valdecoxib (PubChem CID: 119607)
主题词
乙酰胺类(Acetamides);酰胺基水解酶类(Amidohydrolases);动物(Animals);苯并二恶茂类(Benzodioxoles);氨甲酸酯类(Carbamates);环己醇类(Cyclohexanols);环氧化酶2(Cyclooxygenase 2);剂量效应关系, 药物(Dose-Response Relationship, Drug);酶抑制剂(Enzyme Inhibitors);男(雄)性(Male);小鼠, 近交C57BL(Mice, Inbred C57BL);单酰基甘油酯脂酶类(Monoacylglycerol Lipases);哌啶类(Piperidines);吡唑类(Pyrazoles);受体, 大麻酚, CB1(Receptor, Cannabinoid, CB1);琥珀酰亚胺类(Succinimides)
DOI
10.1016/j.neuropharm.2017.06.032
PMID
28673548
发布时间
2019-12-10
- 浏览2
Neuropharmacology
80-86页
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