Platinum(IV) complexes conjugated with phenstatin analogue as inhibitors of microtubule polymerization and reverser of multidrug resistance.
作者:
主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);二苯甲酮类(Benzophenones);结合部位(Binding Sites);细胞系, 肿瘤(Cell Line, Tumor);顺铂(Cisplatin);配位络合物(Coordination Complexes);药物设计(Drug Design);抗药性, 肿瘤(Drug Resistance, Neoplasm);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);人类(Humans);小鼠, 近交BALB C(Mice, Inbred BALB C);小鼠, 裸(Mice, Nude);线粒体(Mitochondria);分子动力学模拟(Molecular Dynamics Simulation);肿瘤(Neoplasms);铂(Platinum);蛋白质结构, 三级(Protein Structure, Tertiary);大鼠(Rats);活性氧(Reactive Oxygen Species);移植, 异种(Transplantation, Heterologous);微管蛋白(Tubulin);微管蛋白调节因子(Tubulin Modulators)
DOI
10.1016/j.bmc.2017.07.011
PMID
28728896
发布时间
2017-12-08
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Bioorganic & medicinal chemistry
4686-4700页
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