Synthesis and pharmacological evaluation of benzamide derivatives as potent and selective sigma-1 protein ligands.

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作者： Marion,Donnier-Maréchal ^[1] ; Pascal,Carato ^[2] ; Paul-Emmanuel,Larchanché ^[3] ; Séverine,Ravez ^[4] ; Rajaa,Boulahjar ^[5] ; Amélie,Barczyk ^[6] ; Bénédicte,Oxombre ^[7] ; Patrick,Vermersch ^[8] ; Patricia,Melnyk ^[9]

作者单位： Univ. Lille, Inserm, CHU Lille, UMR-S 1172 - JPArc - Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, F-59000 Lille, France. Electronic address: md781@cam.ac.uk. ^[1] Univ. Lille, Inserm, CHU Lille, UMR-S 1172 - JPArc - Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, F-59000 Lille, France. Electronic address: pascal.carato@univ-poitiers.fr. ^[2] Univ. Lille, Inserm, CHU Lille, UMR-S 1172 - JPArc - Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, F-59000 Lille, France. Electronic address: paul-emmanuel.larchanche@univ-lille2.fr. ^[3] Univ. Lille, Inserm, CHU Lille, UMR-S 1172 - JPArc - Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, F-59000 Lille, France. Electronic address: severine.ravez@univ-lille2.fr. ^[4] Univ. Lille, Inserm, CHU Lille, UMR-S 1172 - JPArc - Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, F-59000 Lille, France. Electronic address: rajaa.boulahjar@univ-lille2.fr. ^[5] Univ. Lille, Inserm, CHU Lille, U995 - LIRIC - Lille Inflammation Research International Center, F-59000 Lille, France. Electronic address: amelie.barczyk@univ-lille2.fr. ^[6] Univ. Lille, Inserm, CHU Lille, U995 - LIRIC - Lille Inflammation Research International Center, F-59000 Lille, France. Electronic address: benedicte.vanteghem@univ-lille2.fr. ^[7] Univ. Lille, Inserm, CHU Lille, U995 - LIRIC - Lille Inflammation Research International Center, F-59000 Lille, France. Electronic address: patrick.vermersch@univ-lille2.fr. ^[8] Univ. Lille, Inserm, CHU Lille, UMR-S 1172 - JPArc - Centre de Recherche Jean-Pierre AUBERT Neurosciences et Cancer, F-59000 Lille, France. Electronic address: patricia.melnyk@univ-lille2.fr. ^[9]

关键词 Benzamide CNS Sigma protein

主题词苯甲酰胺类(Benzamides);细胞系, 肿瘤(Cell Line, Tumor);剂量效应关系, 药物(Dose-Response Relationship, Drug);人类(Humans);配体(Ligands);分子结构(Molecular Structure);受体, Σ(Receptors, sigma);构效关系(Structure-Activity Relationship)

DOI 10.1016/j.ejmech.2017.07.014

PMID 28756263

发布时间 2017-09-29

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European journal of medicinal chemistry

2017年138卷

964-978页

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Synthesis and pharmacological evaluation of benzamide derivatives as potent and selective sigma-1 protein ligands.

European journal of medicinal chemistry

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European journal of medicinal chemistry

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Synthesis and pharmacological evaluation of benzamide derivatives as potent and selective sigma-1 protein ligands.

European journal of medicinal chemistry

相似文献

European journal of medicinal chemistry

相关期刊

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