Synthesis, enzyme inhibitory kinetics, and computational studies of novel 1-(2-(4-isobutylphenyl) propanoyl)-3-arylthioureas as Jack bean urease inhibitors.
第一作者:
Tanzeela,Abdul Fattah
第一单位:
Department of Chemistry, Quaid-i-Azam University, Islamabad, Pakistan.
作者:
医学主题词
动物(Animals);卤虫属(Artemia);结合部位(Binding Sites);刀豆属(Canavalia);催化域(Catalytic Domain);酶抑制剂(Enzyme Inhibitors);动力学(Kinetics);植物蛋白质类(Plant Proteins);构效关系(Structure-Activity Relationship);热力学(Thermodynamics);硫脲(Thiourea);尿素酶(Urease)
DOI
10.1111/cbdd.13090
PMID
28834266
发布时间
2019-01-25
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Chemical biology & drug design
434-447页
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