PTEN deficiency sensitizes endometrioid endometrial cancer to compound PARP-PI3K inhibition but not PARP inhibition as monotherapy.
第一作者:
X,Bian
第一单位:
Cancer Institute, The Second Hospital of Dalian Medical University, Institute of Cancer Stem Cell, Dalian Medical University, Dalian, China.
作者:
主题词
氨基吡啶类(Aminopyridines);动物(Animals);抗肿瘤联合化疗方案(Antineoplastic Combined Chemotherapy Protocols);癌, 子宫内膜样(Carcinoma, Endometrioid);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);抗药性, 肿瘤(Drug Resistance, Neoplasm);子宫内膜肿瘤(Endometrial Neoplasms);子宫内膜(Endometrium);女(雌)性(Female);人类(Humans);小鼠(Mice);小鼠, 转基因(Mice, Transgenic);吗啉类(Morpholines);肿瘤, 实验性(Neoplasms, Experimental);PTEN磷酸水解酶(PTEN Phosphohydrolase);酞嗪类(Phthalazines);哌嗪类(Piperazines);蛋白激酶抑制剂(Protein Kinase Inhibitors);球形体, 细胞(Spheroids, Cellular)
DOI
10.1038/onc.2017.326
PMID
28945226
发布时间
2019-12-10
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Oncogene
341-351页
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