3'-Hydroxy-3,4'-dimethoxyflavone blocks tubulin polymerization and is a potent apoptotic inducer in human SK-MEL-1 melanoma cells.
作者:
主题词
细胞凋亡(Apoptosis);细胞周期(Cell Cycle);细胞增殖(Cell Proliferation);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);黄酮类(Flavones);人类(Humans);黑色素瘤(Melanoma);显微镜检查, 荧光(Microscopy, Fluorescence);分子结构(Molecular Structure);聚合(Polymerization);构效关系(Structure-Activity Relationship);微管蛋白(Tubulin);肿瘤细胞, 培养的(Tumor Cells, Cultured)
DOI
10.1016/j.bmc.2017.09.043
PMID
29032930
发布时间
2017-12-08
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Bioorganic & medicinal chemistry
6060-6070页
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