A KDM5 Inhibitor Increases Global H3K4 Trimethylation Occupancy and Enhances the Biological Efficacy of 5-Aza-2'-Deoxycytidine.
第一作者:
Benjamin R,Leadem
第一单位:
Department of Oncology, the Sidney Kimmel Comprehensive Cancer Research Center at Johns Hopkins University, Baltimore, Maryland.
作者:
医学主题词
细胞凋亡(Apoptosis);乳腺肿瘤(Breast Neoplasms);细胞增殖(Cell Proliferation);DNA甲基化(DNA Methylation);酶抑制剂(Enzyme Inhibitors);后成说, 遗传(Epigenesis, Genetic);女(雌)性(Female);基因组, 人(Genome, Human);高通量筛选分析(High-Throughput Screening Assays);组蛋白类(Histones);人类(Humans);含Jumonji结构域组蛋白脱甲基酶类(Jumonji Domain-Containing Histone Demethylases);核蛋白质类(Nuclear Proteins);阻遏蛋白质类(Repressor Proteins);肿瘤细胞, 培养的(Tumor Cells, Cultured)
DOI
10.1158/0008-5472.CAN-17-1453
PMID
29282222
发布时间
2019-01-16
- 浏览54
Cancer research
1127-1139页
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