Design, synthesis and biological evaluation of novel bouchardatine analogs as potential inhibitors of adipogenesis/lipogenesis in 3T3-L1 adipocytes.
第一作者:
Lin,Gao
第一单位:
Guangdong Provincial Key Laboratory of New Drug Design and Evaluation, School of Pharmaceutical Sciences, Sun Yat-Sen University, Guangzhou, Guangzhou, 510006, China.
作者:
主题词
3T3-L1细胞(3T3-L1 Cells);脂细胞(Adipocytes);动物(Animals);细胞计数(Cell Count);细胞, 培养的(Cells, Cultured);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物设计(Drug Design);Hep G2细胞(Hep G2 Cells);人类(Humans);吲哚生物碱类(Indole Alkaloids);脂肪生成(Lipogenesis);小鼠(Mice);分子结构(Molecular Structure);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.ejmech.2018.01.089
PMID
29425817
发布时间
2018-03-21
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