Sustained ophthalmic delivery of highly soluble drug using pH-triggered inner layer-embedded contact lens.
第一作者:
Qiang,Zhu
第一单位:
School of Pharmacy, Shenyang Pharmaceutical University, Shenyang 110016, China.
作者:
关键词
2,2′-Azobis(2-methylpropionitrile) (PubChem CID: 6547)2-Hydroxyethyl methacrylate (PubChem CID: 13360)3-Methacryloxypropyl tris (trimethylsiloxy) silane (PubChem CID: 123371)Betaxolol hydrochlorideBetaxolol hydrochloride (PubChem CID: 107952)Ethylene glycol dimethacrylate (PubChem CID: 7355)Extended ocular drug deliveryInner layer-embedded contact lensesMetroprolol succinate (PubChem CID: 62937)N-vinyl-2-pyrrolidone (PubChem CID: 6917)pH-triggered drug release
主题词
肾上腺素能β-1受体拮抗剂(Adrenergic beta-1 Receptor Antagonists);动物(Animals);倍他洛尔(Betaxolol);纤维素(Cellulose);接触镜(Contact Lenses);迟效制剂(Delayed-Action Preparations);药物载体(Drug Carriers);眼(Eye);氢离子浓度(Hydrogen-Ion Concentration);男(雄)性(Male);聚甲基丙烯酸类(Polymethacrylic Acids);兔(Rabbits);溶解度(Solubility)
DOI
10.1016/j.ijpharm.2018.04.004
PMID
29627356
发布时间
2018-09-26
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