Targeting the Proteasome-Associated Deubiquitinating Enzyme USP14 Impairs Melanoma Cell Survival and Overcomes Resistance to MAPK-Targeting Therapies.
第一作者:
Robin,Didier
第一单位:
Inserm, U1065, Team Microenvironment, Signaling and Cancer, Centre Méditerranéen de Médecine Moléculaire (C3M) and Université Côte d'Azur, Nice, France.;Equipe labellisée Ligue Contre le Cancer 2016, Nice, France.
作者:
医学主题词
动物(Animals);细胞凋亡(Apoptosis);细胞系, 肿瘤(Cell Line, Tumor);细胞存活(Cell Survival);抗药性, 肿瘤(Drug Resistance, Neoplasm);GTP磷酸水解酶类(GTP Phosphohydrolases);基因表达调控, 肿瘤(Gene Expression Regulation, Neoplastic);人类(Humans);MAP激酶激酶1(MAP Kinase Kinase 1);黑素细胞(Melanocytes);黑色素瘤(Melanoma);膜蛋白质类(Membrane Proteins);小鼠(Mice);分子靶向治疗(Molecular Targeted Therapy);原癌基因蛋白质B-raf(Proto-Oncogene Proteins B-raf);活性氧(Reactive Oxygen Species);肿瘤抑制蛋白质p53(Tumor Suppressor Protein p53);泛素硫酯酶(Ubiquitin Thiolesterase);异种移植模型抗肿瘤试验(Xenograft Model Antitumor Assays)
DOI
10.1158/1535-7163.MCT-17-0919
PMID
29703842
发布时间
2020-09-30
- 浏览15
Molecular cancer therapeutics
1416-1429页
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