Synthesis and Biological in vitro and in vivo Evaluation of 2-(5-Nitroindazol-1-yl)ethylamines and Related Compounds as Potential Therapeutic Alternatives for Chagas Disease.
第一作者:
Rubén,Martín-Escolano
第一单位:
Department of Parasitology, Instituto de Investigación Biosanitaria (ibs.Granada), Hospitales Universitarios de Granada, University of Granada, c/ Severo Ochoa s/n, 18071, Granada, Spain.
作者:
主题词
动物(Animals);Chagas病(Chagas Disease);DNA(DNA);酶抑制剂(Enzyme Inhibitors);乙胺类(Ethylamines);女(雌)性(Female);吲唑类(Indazoles);膜电位, 线粒体(Membrane Potential, Mitochondrial);小鼠, 近交BALB C(Mice, Inbred BALB C);被忽略疾病(Neglected Diseases);RNA(RNA);超氧化物歧化酶(Superoxide Dismutase);抗锥虫药(Trypanocidal Agents);克鲁斯锥虫(Trypanosoma cruzi);Vero细胞(Vero Cells)
DOI
10.1002/cmdc.201800512
PMID
30098232
发布时间
2019-12-10
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ChemMedChem
2104-2118页
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