Design and development of novel p-aminobenzoic acid derivatives as potential cholinesterase inhibitors for the treatment of Alzheimer's disease.
第一作者:
Sushant K,Shrivastava
第一单位:
Pharmaceutical Chemistry Research Laboratory, Department of Pharmaceutical Engineering & Technology, Indian Institute of Technology (Banaras Hindu University), Varanasi 221005, U.P., India. Electronic address: skshrivastava.phe@iitbhu.ac.in.
作者:
医学主题词
乙酰胆碱酯酶(Acetylcholinesterase);阿尔茨海默病(Alzheimer Disease);动物(Animals);脑(Brain);丁酰胆碱酯酶(Butyrylcholinesterase);催化域(Catalytic Domain);胆碱酯酶抑制剂(Cholinesterase Inhibitors);药物设计(Drug Design);女(雌)性(Female);动力学(Kinetics);男(雄)性(Male);记忆(Memory);分子动力学模拟(Molecular Dynamics Simulation);分子结构(Molecular Structure);脑代谢改善药(Nootropic Agents);量化构效关系(Quantitative Structure-Activity Relationship);大鼠(Rats);缩氨基脲类(Semicarbazones)
DOI
10.1016/j.bioorg.2018.10.009
PMID
30326403
发布时间
2019-08-30
- 浏览14
Bioorganic chemistry
211-223页
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