Synthesis, biological evaluation and molecular dynamic simulations of novel Benzofuran-tetrazole derivatives as potential agents against Alzheimer's disease.
作者:
主题词
乙酰胆碱酯酶(Acetylcholinesterase);阿尔茨海默病(Alzheimer Disease);淀粉样β肽类(Amyloid beta-Peptides);动物(Animals);苯呋喃类(Benzofurans);秀丽新小杆线虫(Caenorhabditis elegans);胆碱酯酶抑制剂(Cholinesterase Inhibitors);剂量效应关系, 药物(Dose-Response Relationship, Drug);分子动力学模拟(Molecular Dynamics Simulation);分子结构(Molecular Structure);构效关系(Structure-Activity Relationship);四唑类(Tetrazoles)
DOI
10.1016/j.bmcl.2018.11.005
PMID
30455151
发布时间
2019-11-04
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