Capmatinib (INC280) Is Active Against Models of Non-Small Cell Lung Cancer and Other Cancer Types with Defined Mechanisms of MET Activation.
第一作者:
Sabrina,Baltschukat
第一单位:
Novartis Institutes for BioMedical Research, Oncology Disease Area, Basel, Switzerland.
作者:
主题词
动物(Animals);苯甲酰胺类(Benzamides);癌, 非小细胞肺(Carcinoma, Non-Small-Cell Lung);细胞系, 肿瘤(Cell Line, Tumor);药物评价, 临床前(Drug Evaluation, Preclinical);抗药性, 肿瘤(Drug Resistance, Neoplasm);酶激活(Enzyme Activation);胶质母细胞瘤(Glioblastoma);肝细胞生长因子(Hepatocyte Growth Factor);人类(Humans);咪唑类(Imidazoles);肺肿瘤(Lung Neoplasms);小鼠(Mice);蛋白激酶抑制剂(Protein Kinase Inhibitors);原癌基因蛋白质c-met(Proto-Oncogene Proteins c-met);胃肿瘤(Stomach Neoplasms);三嗪类(Triazines);异种移植模型抗肿瘤试验(Xenograft Model Antitumor Assays)
DOI
10.1158/1078-0432.CCR-18-2814
PMID
30674502
发布时间
2021-12-04
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Clinical cancer research
3164-3175页
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