Structural Basis of Altered Potency and Efficacy Displayed by a Major in Vivo Metabolite of the Antidiabetic PPARγ Drug Pioglitazone.
第一作者:
Sarah A,Mosure
第一单位:
Department of Integrative Structural and Computational Biology , The Scripps Research Institute , La Jolla , California 92037 , United States.
作者:
主题词
结合部位(Binding Sites);HEK293细胞(HEK293 Cells);人类(Humans);氢键合(Hydrogen Bonding);降血糖药(Hypoglycemic Agents);PPARγ(PPAR gamma);蛋白质结合(Protein Binding);蛋白质构象(Protein Conformation);立体异构现象(Stereoisomerism)
DOI
10.1021/acs.jmedchem.8b01573
PMID
30676741
发布时间
2023-04-15
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Journal of medicinal chemistry
2008-2023页
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