Design and development of 1,3,4-oxadiazole derivatives as potential inhibitors of acetylcholinesterase to ameliorate scopolamine-induced cognitive dysfunctions.
第一作者:
Puja,Mishra
第一单位:
Department of Pharmaceutical Engineering & Technology, Indian Institute of Technology (Banaras Hindu University), Varanasi 221 005, India.
作者:
医学主题词
乙酰胆碱酯酶(Acetylcholinesterase);淀粉样β肽类(Amyloid beta-Peptides);动物(Animals);回避学习(Avoidance Learning);丁酰胆碱酯酶(Butyrylcholinesterase);胆碱酯酶抑制剂(Cholinesterase Inhibitors);剂量效应关系, 药物(Dose-Response Relationship, Drug);电鳗属(Electrophorus);马(Horses);人类(Humans);男(雄)性(Male);记忆(Memory);小鼠(Mice);分子结构(Molecular Structure);恶二唑类(Oxadiazoles);肽碎片(Peptide Fragments);氢溴酸东莨菪碱(Scopolamine Hydrobromide);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bioorg.2019.103025
PMID
31176239
发布时间
2020-09-22
- 浏览0
Bioorganic chemistry
103025页
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