Discovery of 4<i>H</i>-Chromen-4-one Derivatives as a New Class of Selective Rho Kinase (ROCK) Inhibitors, which Showed Potent Activity in ex Vivo Diabetic Retinopathy Models.
作者:
主题词
动物(Animals);糖尿病视网膜病变(Diabetic Retinopathy);药物发现(Drug Discovery);葡萄糖(Glucose);人类(Humans);小鼠(Mice);小鼠, 近交C57BL(Mice, Inbred C57BL);蛋白激酶抑制剂(Protein Kinase Inhibitors);组织培养技术(Tissue Culture Techniques);rho相关激酶类(rho-Associated Kinases)
DOI
10.1021/acs.jmedchem.9b01143
PMID
31693351
发布时间
2020-06-22
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Journal of medicinal chemistry
10691-10710页
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