Meeting organometallic chemistry with drug discovery: CH activation enabled discovery of a new ring system of 12H-Indazolo[2,1-a]cinnolin-12-ones with anti-proliferation activity.
作者:
主题词
烷化作用(Alkylation);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);碳(Carbon);半胱氨酸天冬氨酸蛋白酶3(Caspase 3);催化作用(Catalysis);细胞系, 肿瘤(Cell Line, Tumor);细胞存活(Cell Survival);药物设计(Drug Design);杂环化合物, 2环(Heterocyclic Compounds, 2-Ring);人类(Humans);氢(Hydrogen);有机金属化合物(Organometallic Compounds);铑(Rhodium);钌化合物(Ruthenium Compounds);增量调节(Up-Regulation)
DOI
10.1016/j.bmcl.2019.126916
PMID
31889668
发布时间
2021-01-28
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