Aminotriazines with indole motif as novel, 5-HT<sub>7</sub> receptor ligands with atypical binding mode.
第一作者:
Damian,Kułaga
第一单位:
Faculty of Chemical Engineering and Technology, Institute of Organic Chemistry and Technology, Cracow University of Technology, 24 Warszawska Street, 31-155 Kraków, Poland. Electronic address: damian.kulaga@doktorant.pk.edu.pl.
作者:
医学主题词
结合部位(Binding Sites);剂量效应关系, 药物(Dose-Response Relationship, Drug);Hep G2细胞(Hep G2 Cells);人类(Humans);吲哚类(Indoles);配体(Ligands);模型, 分子(Models, Molecular);分子结构(Molecular Structure);受体, 血清素(Receptors, Serotonin);血清素拮抗药(Serotonin Antagonists);血清素受体激动剂(Serotonin Receptor Agonists);构效关系(Structure-Activity Relationship);三嗪类(Triazines)
DOI
10.1016/j.bioorg.2020.104254
PMID
32919133
发布时间
2021-03-29
- 浏览0
Bioorganic chemistry
104254页
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