Synthesis, ADMET prediction and reverse screening study of 3,4,5-trimethoxy phenyl ring pendant sulfur-containing cyanopyrimidine derivatives as promising apoptosis inducing anticancer agents.
第一作者:
Lalit Mohan,Nainwal
第一单位:
Drug Design & Medicinal Chemistry Lab, Department of Pharmaceutical Chemistry, School of Pharmaceutical Education and Research, Jamia Hamdard, New Delhi 110062, India.
作者:
医学主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);狗(Dogs);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物评价, 临床前(Drug Evaluation, Preclinical);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);人类(Humans);分子结构(Molecular Structure);嘧啶类(Pyrimidines);构效关系(Structure-Activity Relationship);硫(Sulfur)
DOI
10.1016/j.bioorg.2020.104282
PMID
33010624
发布时间
2021-03-29
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Bioorganic chemistry
104282页
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