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The IMiD target CRBN determines HSP90 activity toward transmembrane proteins essential in multiple myeloma.

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作者单位: Department of Medicine III, Klinikum rechts der Isar, Technical University of Munich, 81675 Munich, Germany; TranslaTUM, Center for Translational Cancer Research, Technical University of Munich, 81675 Munich, Germany. [1] Department of Nuclear Medicine, Klinikum rechts der Isar, Technical University of Munich, 81675 Munich, Germany. [2] Department of Proteomics and Bioanalytics, Technical University of Munich, 85354 Freising, Germany; German Cancer Consortium (DKTK) and German Cancer Research Center (DKFZ), 69120 Heidelberg, Germany. [3] Center for Integrated Protein Science at the Department of Chemistry, Technical University of Munich, 85748 Garching, Germany. [4] Department of Molecular Machines and Signaling, Max Planck Institute of Biochemistry, 82152 Martinsried, Germany. [5] Department of Medicine III, Klinikum rechts der Isar, Technical University of Munich, 81675 Munich, Germany. [6] Institute of Pathology, Ludwig-Maximilians University, 80337 Munich, Germany. [7] Lehrstuhl für Biologische Chemie, Technical University of Munich, 85354 Freising, Germany. [8] German Cancer Consortium (DKTK) and German Cancer Research Center (DKFZ), 69120 Heidelberg, Germany; Department of Hematology, Oncology and Tumor Immunology (Campus Benjamin Franklin), Charité - Universitätsmedizin Berlin, 12200 Berlin, Germany. [9] Department of Proteomics and Bioanalytics, Technical University of Munich, 85354 Freising, Germany. [10] Department of Medicine III, Klinikum rechts der Isar, Technical University of Munich, 81675 Munich, Germany; German Cancer Consortium (DKTK) and German Cancer Research Center (DKFZ), 69120 Heidelberg, Germany. [11] Department of Nuclear Medicine, Klinikum rechts der Isar, Technical University of Munich, 81675 Munich, Germany; German Cancer Consortium (DKTK) and German Cancer Research Center (DKFZ), 69120 Heidelberg, Germany. [12] Department of Medicine III, Klinikum rechts der Isar, Technical University of Munich, 81675 Munich, Germany; TranslaTUM, Center for Translational Cancer Research, Technical University of Munich, 81675 Munich, Germany. Electronic address: vanesa.fernandez@tum.de. [13] Department of Medicine III, Klinikum rechts der Isar, Technical University of Munich, 81675 Munich, Germany; TranslaTUM, Center for Translational Cancer Research, Technical University of Munich, 81675 Munich, Germany; German Cancer Consortium (DKTK) and German Cancer Research Center (DKFZ), 69120 Heidelberg, Germany. Electronic address: florian.bassermann@tum.de. [14]
DOI 10.1016/j.molcel.2020.12.046
PMID 33571422
发布时间 2021-04-01
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Molecular cell

Molecular cell

2021年81卷6期

1170-1186.e10页

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