Identification of NSAIDs as lipoxygenase inhibitors through highly sensitive chemiluminescence method, expression analysis in mononuclear cells and computational studies.
第一作者:
Wardah,Shahid
第一单位:
Department of Chemistry, The Islamia University of Bahawalpur, Bahawalpur 63100, Pakistan.
作者:
医学主题词
消炎药, 非甾类(Anti-Inflammatory Agents, Non-Steroidal);花生四烯酸盐15-脂氧合酶(Arachidonate 15-Lipoxygenase);花生四烯酸盐5-脂氧合酶(Arachidonate 5-Lipoxygenase);剂量效应关系, 药物(Dose-Response Relationship, Drug);人类(Humans);脂氧合酶抑制剂(Lipoxygenase Inhibitors);发光测定法(Luminescent Measurements);分子结构(Molecular Structure);构效关系(Structure-Activity Relationship)
DOI
10.1016/j.bioorg.2021.104818
PMID
33784531
发布时间
2021-10-12
- 浏览0
Bioorganic chemistry
104818页
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