From High-Throughput Screening to Target Validation: Benzo[<i>d</i>]isothiazoles as Potent and Selective Agonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 5 Possessing In Vivo Gastrointestinal Prokinetic Activity in Rodents.
第一作者:
Alessio,Barilli
第一单位:
Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
作者:
医学主题词
动物(Animals);苯并噻唑类(Benzothiazoles);药物设计(Drug Design);胃肠道(Gastrointestinal Tract);高通量筛选分析(High-Throughput Screening Assays);人类(Humans);男(雄)性(Male);小鼠(Mice);分子靶向治疗(Molecular Targeted Therapy);结果可重复性(Reproducibility of Results);TRPM阳离子通道(TRPM Cation Channels);组织分布(Tissue Distribution)
DOI
10.1021/acs.jmedchem.1c00065
PMID
33890770
发布时间
2021-06-14
- 浏览2
Journal of medicinal chemistry
5931-5955页
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