Discovery of an H3K36me3-Derived Peptidomimetic Ligand with Enhanced Affinity for Plant Homeodomain Finger Protein 1 (PHF1).
第一作者:
Isabelle A,Engelberg
第一单位:
Center for Integrative Chemical Biology and Drug Discovery, Division of Chemical Biology and Medicinal Chemistry, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina 27599, United States.
作者:
主题词
氨基酸序列(Amino Acid Sequence);结晶学, X线(Crystallography, X-Ray);DNA结合蛋白质类(DNA-Binding Proteins);人类(Humans);配体(Ligands);诱变, 定点(Mutagenesis, Site-Directed);核磁共振, 生物分子(Nuclear Magnetic Resonance, Biomolecular);多肽模拟物(Peptidomimetics);蛋白质结合(Protein Binding)
DOI
10.1021/acs.jmedchem.1c00430
PMID
33999620
发布时间
2022-07-16
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Journal of medicinal chemistry
8510-8522页
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