Design, Synthesis, and Activity Evaluation of Stereoconfigured Tartarate Derivatives as Potential Anti-inflammatory Agents <i>In Vitro</i> and <i>In Vivo</i>.
作者:
主题词
动物(Animals);消炎药, 非甾类(Anti-Inflammatory Agents, Non-Steroidal);角叉菜胶(Carrageenan);环氧化酶2(Cyclooxygenase 2);环氧化酶2抑制剂(Cyclooxygenase 2 Inhibitors);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物设计(Drug Design);水肿(Edema);女(雌)性(Female);人类(Humans);脂氧合酶(Lipoxygenase);脂氧合酶抑制剂(Lipoxygenase Inhibitors);男(雄)性(Male);小鼠(Mice);分子结构(Molecular Structure);立体异构现象(Stereoisomerism);构效关系(Structure-Activity Relationship);酒石酸盐类(Tartrates)
DOI
10.1021/acs.jmedchem.1c00880
PMID
34137625
发布时间
2021-09-07
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Journal of medicinal chemistry
9550-9566页
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