Asymmetric Synthesis and Biological Screening of Quinoxaline-Containing Synthetic Lipoxin A<sub>4</sub> Mimetics (QNX-sLXms).
第一作者:
Monica,de Gaetano
第一单位:
School of Medicine, Diabetes Complications Research Centre, UCD Conway Institute, University College Dublin, Belfield, Dublin D04 N2E5, Ireland.
作者:
主题词
动物(Animals);消炎药, 非甾类(Anti-Inflammatory Agents, Non-Steroidal);细胞存活(Cell Survival);细胞, 培养的(Cells, Cultured);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物评价, 临床前(Drug Evaluation, Preclinical);人类(Humans);炎症(Inflammation);脂多糖类(Lipopolysaccharides);小鼠(Mice);分子结构(Molecular Structure);单核细胞(Monocytes);NF-κB(NF-kappa B);喹恶啉类(Quinoxalines);受体, 甲酰肽(Receptors, Formyl Peptide);受体, 脂氧素(Receptors, Lipoxin);构效关系(Structure-Activity Relationship);肿瘤坏死因子α(Tumor Necrosis Factor-alpha)
DOI
10.1021/acs.jmedchem.1c00403
PMID
34138563
发布时间
2021-09-07
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Journal of medicinal chemistry
9193-9216页
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