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Molecular insights into ago-allosteric modulation of the human glucagon-like peptide-1 receptor.

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作者: Zhaotong,Cong [1] ; Li-Nan,Chen [2] ; Honglei,Ma [3] ; Qingtong,Zhou [2] ; Xinyu,Zou [4] ; Chenyu,Ye [5] ; Antao,Dai [1] ; Qing,Liu [2] ; Wei,Huang [6] ; Xianqiang,Sun [6] ; Xi,Wang [7] ; Peiyu,Xu [7] ; Lihua,Zhao [2] ; Tian,Xia [8] ; Wenge,Zhong [2] ; Dehua,Yang [2] ; H,Eric Xu [5] ; Yan,Zhang [7] ; Ming-Wei,Wang [9]
作者单位: School of Pharmacy, Fudan University, Shanghai, China. [1] The CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China. [2] Department of Biophysics and Department of Pathology of Sir Run Run Shaw Hospital, Zhejiang University School of Medicine, Hangzhou, China. [3] School of Basic Medical Sciences, Fudan University, Shanghai, China. [4] School of Artificial Intelligence and Automation, Huazhong University of Science and Technology, Wuhan, China. [5] The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China. [6] Qilu Regor Therapeutics, Inc., Shanghai, China. [7] University of Chinese Academy of Sciences, Beijing, China. [8] The CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China. dhyang@simm.ac.cn. [9] The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China. dhyang@simm.ac.cn. [10] University of Chinese Academy of Sciences, Beijing, China. dhyang@simm.ac.cn. [11] The CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China. eric.xu@simm.ac.cn. [12] University of Chinese Academy of Sciences, Beijing, China. eric.xu@simm.ac.cn. [13] Department of Biophysics and Department of Pathology of Sir Run Run Shaw Hospital, Zhejiang University School of Medicine, Hangzhou, China. zhang_yan@zju.edu.cn. [14] MOE Frontier Science Center for Brain Research and Brain-Machine Integration, Zhejiang University School of Medicine, Hangzhou, China. zhang_yan@zju.edu.cn. [15] Key Laboratory of Immunity and Inflammatory Diseases of Zhejiang Province, Hangzhou, China. zhang_yan@zju.edu.cn. [16] Zhejiang Laboratory for Systems and Precision Medicine, Zhejiang University Medical Center, Hangzhou, China. zhang_yan@zju.edu.cn. [17] School of Life Science and Technology, ShanghaiTech University, Shanghai, China. zhang_yan@zju.edu.cn. [18] School of Pharmacy, Fudan University, Shanghai, China. mwwang@simm.ac.cn. [19] The CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China. mwwang@simm.ac.cn. [20] School of Basic Medical Sciences, Fudan University, Shanghai, China. mwwang@simm.ac.cn. [21] The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China. mwwang@simm.ac.cn. [22] University of Chinese Academy of Sciences, Beijing, China. mwwang@simm.ac.cn. [23] School of Life Science and Technology, ShanghaiTech University, Shanghai, China. mwwang@simm.ac.cn. [24]
DOI 10.1038/s41467-021-24058-z
PMID 34145245
发布时间 2021-07-06
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