Synthesis and Biological Evaluation of C-17-Amino-Substituted Pyrazole-Fused Betulinic Acid Derivatives as Novel Agents for Osteoarthritis Treatment.
第一作者:
Jie,Wang
第一单位:
State Key Laboratory of Drug Research, Department of Medicinal Chemistry, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai 201203, China.
作者:
主题词
动物(Animals);消炎药(Anti-Inflammatory Agents);骨和骨组织(Bone and Bones);软骨, 关节(Cartilage, Articular);细胞分化(Cell Differentiation);碘乙酸(Iodoacetic Acid);脂多糖类(Lipopolysaccharides);巨噬细胞集落刺激因子(Macrophage Colony-Stimulating Factor);男(雄)性(Male);小鼠(Mice);骨关节炎(Osteoarthritis);破骨细胞(Osteoclasts);五环三萜类(Pentacyclic Triterpenes);吡唑类(Pyrazoles);RANK配体(RANK Ligand);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);大鼠(Rats)
DOI
10.1021/acs.jmedchem.1c01019
PMID
34491054
发布时间
2024-02-26
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Journal of medicinal chemistry
13676-13692页
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