A Glutamate <i>N</i>-Methyl-d-Aspartate (NMDA) Receptor Subunit 2B-Selective Inhibitor of NMDA Receptor Function with Enhanced Potency at Acidic pH and Oral Bioavailability for Clinical Use.
第一作者:
Scott J,Myers
第一单位:
Department of Pharmacology and Chemical Biology (S.J.M, P.L., R.J.D., S.F.T.), Department of Chemistry (L.J.W., Y.A.T., D.S.M., Z.W.D., D.C.L.), Emory University, Atlanta, Georgia; NeurOp Inc., Atlanta, Georgia (S.J.M., K.P.R., L.J.W., Y.A.T, P.L., D.S.M., Z.W.D., G.W.K., R.Z.), and TRPblue Inc., Durham, North Carolina (G.W.K).
作者:
主题词
酸类(Acids);投药, 口服(Administration, Oral);动物(Animals);生物利用度(Biological Availability);脑(Brain);剂量效应关系, 药物(Dose-Response Relationship, Drug);兴奋性氨基酸拮抗剂(Excitatory Amino Acid Antagonists);女(雌)性(Female);氢离子浓度(Hydrogen-Ion Concentration);男(雄)性(Male);小鼠(Mice);小鼠, 近交C57BL(Mice, Inbred C57BL);受体, N-甲基-D-天冬氨酸(Receptors, N-Methyl-D-Aspartate);光滑爪蟾(Xenopus laevis)
DOI
10.1124/jpet.120.000370
PMID
34493631
发布时间
2025-03-06
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