Discovery of Novel Histone Deacetylase 6 (HDAC6) Inhibitors with Enhanced Antitumor Immunity of Anti-PD-L1 Immunotherapy in Melanoma.
作者:
主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);药物协同作用(Drug Synergism);组蛋白脱乙酰基酶抑制剂(Histone Deacetylase Inhibitors);人类(Humans);羟肟酸类(Hydroxamic Acids);免疫(Immunity);免疫疗法(Immunotherapy);男(雄)性(Male);黑色素瘤(Melanoma);小鼠(Mice);分子结构(Molecular Structure);大鼠, Sprague-Dawley(Rats, Sprague-Dawley);构效关系(Structure-Activity Relationship);噻唑类(Thiazoles);大鼠(Rats)
DOI
10.1021/acs.jmedchem.1c01863
PMID
35043615
发布时间
2024-10-19
- 浏览5

Journal of medicinal chemistry
2434-2457页
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