Angiogenesis and anti-leukaemia activity of novel indole derivatives as potent colchicine binding site inhibitors.
作者:
主题词
血管生成抑制剂(Angiogenesis Inhibitors);动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞凋亡(Apoptosis);结合部位(Binding Sites);细胞系, 肿瘤(Cell Line, Tumor);细胞增殖(Cell Proliferation);秋水仙碱(Colchicine);剂量效应关系, 药物(Dose-Response Relationship, Drug);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);人类(Humans);吲哚类(Indoles);模型, 分子(Models, Molecular);分子结构(Molecular Structure);肿瘤, 实验性(Neoplasms, Experimental);新生血管化, 病理性(Neovascularization, Pathologic);构效关系(Structure-Activity Relationship);微管蛋白(Tubulin);微管蛋白调节因子(Tubulin Modulators);斑马鱼(Zebrafish)
DOI
10.1080/14756366.2022.2032688
PMID
35109719
发布时间
2022-03-21
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