Structure-Activity Relationship Study of Indolin-5-yl-cyclopropanamine Derivatives as Selective Lysine Specific Demethylase 1 (LSD1) Inhibitors.
第一作者:
Chunpu,Li
第一单位:
State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.
作者:
主题词
动物(Animals);抗肿瘤药(Antineoplastic Agents);细胞增殖(Cell Proliferation);酶抑制剂(Enzyme Inhibitors);组蛋白脱甲基酶类(Histone Demethylases);人类(Humans);吲哚类(Indoles);白血病, 髓样, 急性(Leukemia, Myeloid, Acute);赖氨酸(Lysine);小鼠(Mice);构效关系(Structure-Activity Relationship)
DOI
10.1021/acs.jmedchem.1c02156
PMID
35200034
发布时间
2022-05-06
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Journal of medicinal chemistry
4335-4349页
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