Compounds targeting GPI biosynthesis or <i>N</i>-glycosylation are active against <i>Plasmodium falciparum</i>.
第一作者:
Àngel,Fenollar
第一单位:
Barcelona Institute for Global Health (ISGlobal), Hospital Clínic-University of Barcelona, 08036 Barcelona, Spain.
作者:
关键词
ALG7, UDP-N-acetylglucosamine:dolichyl-phosphateN-acetylglucosaminephosphotransferaseAntiplasmodial activityCDS, Coding sequenceCSP, Circumsporozoite proteinDMSO, Dimethyl sulfoxideER, Endoplasmic reticulumGPI, GlycosylphosphatidylinositolGPI-anchorsGSL-II, Griffonia simplicifoliaII lectinGWT1, Inositol acyltransferaseGlcNAc, N-acetylglucosamineGlcNAc-PI de-N-acetylase, N-acetylglucosaminyl-phosphatidylinositol de-N-acetylaseIDC, Intraerythrocytic developmental cycleInhibitorsMalariaN-glycans, Asparagine-linked glycansN-glycosylationOST, OligosaccharyltransferasePlasmodium falciparumRBCs, Red blood cellsSHAM, Salicylic hydroxamic acidUDP-GlcNAc, UDP-N-acetylglucosaminepLDDT, Predicted local distance difference test
DOI
10.1016/j.csbj.2022.01.029
PMID
35222844
发布时间
2022-03-01
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