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Clinical evaluation of [<sup>18</sup>F]pitavastatin for quantitative analysis of hepatobiliary transporter activity.

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作者单位: RIKEN Center for Life Science Technologies CLST, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan; RIKEN Center for Biosystems Dynamics Research BDR, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan. [1] RIKEN Center for Life Science Technologies CLST, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan. [2] RIKEN Center for Biosystems Dynamics Research BDR, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan. [3] Department of Physiology, Graduate School of Medicine, Osaka City University, Abeno-ku, Osaka, 545-8585, Japan. [4] Department of Hepatology, Graduate School of Medicine, Osaka City University, Abeno-ku, Osaka, 545-8585, Japan. [5] Department of Radiology, Osaka City University Hospital, Abeno-ku, Osaka, 545-8586, Japan. [6] Department of Nuclear Medicine, Graduate School of Medicine, Osaka City University, Abeno-ku, Osaka, 545-8585, Japan. [7] Department of Diagnostic and Interventional Radiology, Graduate School of Medicine, Osaka City University, Abeno-ku, Osaka, 545-8585, Japan. [8] RIKEN Center for Life Science Technologies CLST, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan; RIKEN Center for Biosystems Dynamics Research BDR, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan; Laboratory of Chemical Bioscience, Institute of Biomaterials and Bioengineering, Tokyo Medical and Dental University TMDU, 2-3-10 Kanda-Surugadai, Chiyoda-ku, Tokyo, 101-0062, Japan. [9] Laboratory of Molecular Pharmacokinetics, Graduate School of Pharmaceutical Sciences, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo, 113-0033, Japan; Kitasato University School of Pharmacy, 5-9-1 Shirokane, Minato-ku, Tokyo, 108-8641, Japan. [10] Laboratory of Molecular Pharmacokinetics, Graduate School of Pharmaceutical Sciences, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo, 113-0033, Japan. [11] Sugiyama Laboratory, RIKEN Innovation Center, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama, Kanagawa, 230-0045, Japan; Laboratory of Quantitative System Pharmacokinetics / Pharmacodynamics, School of Pharmacy, Josai International University, Kioi-cho, Tokyo, 102-0093, Japan. [12] RIKEN Center for Life Science Technologies CLST, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan; RIKEN Center for Biosystems Dynamics Research BDR, 6-7-3 Minatojima-minamimachi, Chuo-ku, Kobe, Hyogo, 650-0047, Japan. Electronic address: yywata@riken.jp. [13]
DOI 10.1016/j.dmpk.2022.100449
PMID 35395593
发布时间 2022-06-02
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