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Comprehensive Fragment Screening of the SARS-CoV-2 Proteome Explores Novel Chemical Space for Drug Development.

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作者: Hannes,Berg [1] ; Maria A,Wirtz Martin [2] ; Nadide,Altincekic [1] ; Islam,Alshamleh [2] ; Jasleen,Kaur Bains [1] ; Julius,Blechar [2] ; Betül,Ceylan [1] ; Vanessa,de Jesus [2] ; Karthikeyan,Dhamotharan [1] ; Christin,Fuks [2] ; Santosh L,Gande [1] ; Bruno,Hargittay [1] ; Katharina F,Hohmann [2] ; Marie T,Hutchison [1] ; Sophie,Marianne Korn [2] ; Robin,Krishnathas [2] ; Felicitas,Kutz [3] ; Verena,Linhard [1] ; Tobias,Matzel [1] ; Nathalie,Meiser [2] ; Anna,Niesteruk [1] ; Dennis J,Pyper [2] ; Linda,Schulte [1] ; Sven,Trucks [2] ; Kamal,Azzaoui [1] ; Marcel J J,Blommers [2] ; Yojana,Gadiya [2] ; Reagon,Karki [3] ; Andrea,Zaliani [1] ; Philip,Gribbon [2] ; Marcius,da Silva Almeida [1] ; Cristiane,Dinis Anobom [2] ; Anna L,Bula [1] ; Matthias,Bütikofer [2] ; Ícaro,Putinhon Caruso [1] ; Isabella,Caterina Felli [2] ; Andrea T,Da Poian [1] ; Gisele,Cardoso de Amorim [1] ; Nikolaos K,Fourkiotis [2] ; Angelo,Gallo [1] ; Dhiman,Ghosh [2] ; Francisco,Gomes-Neto [1] ; Oksana,Gorbatyuk [2] ; Bing,Hao [1] ; Vilius,Kurauskas [4] ; Lauriane,Lecoq [4] ; Yunfeng,Li [5] ; Nathane,Cunha Mebus-Antunes [6] ; Miguel,Mompeán [5] ; Thais,Cristtina Neves-Martins [6] ; Martí,Ninot-Pedrosa [5] ; Anderson S,Pinheiro [6] ; Letizia,Pontoriero [5] ; Yulia,Pustovalova [6] ; Roland,Riek [7] ; Angus J,Robertson [6] ; Marie,Jose Abi Saad [8] ; Miguel Á,Treviño [9] ; Aikaterini C,Tsika [10] ; Fabio C L,Almeida [11] ; Ad,Bax [7] ; Katherine,Henzler-Wildman [12] ; Jeffrey C,Hoch [13] ; Kristaps,Jaudzems [14] ; Douglas V,Laurents [7] ; Julien,Orts [7] ; Roberta,Pierattelli [15] ; Georgios A,Spyroulias [16] ; Elke,Duchardt-Ferner [16] ; Jan,Ferner [17] ; Boris,Fürtig [11] ; Martin,Hengesbach [8] ; Frank,Löhr [18] ; Nusrat,Qureshi [19] ; Christian,Richter [19] ; Krishna,Saxena [20] ; Andreas,Schlundt [21] ; Sridhar,Sreeramulu [19] ; Anna,Wacker [7] ; Julia E,Weigand [22] ; Julia,Wirmer-Bartoschek [7] ; Jens,Wöhnert [21] ; Harald,Schwalbe [9]
作者单位: Institute for Organic Chemistry and Chemical Biology, Goethe University Frankfurt, 60438, Frankfurt am Main, Germany. [1] Center of Biomolecular Magnetic Resonance (BMRZ), Goethe University Frankfurt, Frankfurt am Main (Germany), Max-von-LaueStrasse 7+9, 60438, Frankfurt am Main, Germany. [2] Institute for Molecular Biosciences, Goethe University Frankfurt, Max-von-Laue Strasse 7+9, 60438, Frankfurt am Main, Germany. [3] Saverna Therapeutics, Pumpmattenweg 3, 4105, Biel-Benken, Switzerland. [4] Fraunhofer Institute for Translational Medicine and Pharmacology (ITMP), Screening Port, Schnackenburgallee 114, 22525, Hamburg, Germany. [5] Fraunhofer Cluster of Excellence for Immune-Mediated Diseases (CIMD), Theodor-Stern-Kai 7, 60596, Frankfurt am Main, Germany. [6] Institute of Medical Biochemistry, Federal University of Rio de Janeiro, 21941-902, Rio de Janeiro, Brazil. [7] National Center of Nuclear Magnetic Resonance (CNRMN), CENABIO, Federal University of Rio de Janeiro, 21941-902, Rio de Janeiro, Brazil. [8] Department of Biochemistry, Institute of Chemistry, Federal University of Rio de Janeiro, 21941-902, Rio de Janeiro, Brazil. [9] Latvian Institute of Organic Synthesis, Aizkraukles 21, LV-1006, Riga, Latvia. [10] ETH, Swiss Federal Institute of Technology, Laboratory of Physical Chemistry, HCI F217, Vladimir-Prelog-Weg 2, 8093, Zürich, Switzerland. [11] Multiuser Center for Biomolecular Innovation (CMIB), Department of Physics, São Paulo State University (UNESP), 01049-010, São José do Rio Preto, Brazil. [12] Magnetic Resonance Center (CERM), University of Florence, Via Luigi Sacconi 6, Sesto Fiorentino, 50019, Florence, Italy. [13] Department of Chemistry "Ugo Schiff", University of Florence, Via della Lastruccia 3-13, Sesto Fiorentino, 50019, Florence, Italy. [14] Multidisciplinary Center for Research in Biology (NUMPEX), Campus Duque de Caxias Federal University of Rio de Janeiro, 25.250-470, Duque de Caxias, Brazil. [15] Department of Pharmacy, University of Patras, 26504, Patras, Greece. [16] Department of Chemistry, University of Torino, IT-10126, Torino, Italy. [17] Laboratory of Toxinology, Oswaldo Cruz Foundation (FIOCRUZ), 21040-900, Rio de Janeiro, Brazil. [18] Department of Molecular Biology and Biophysics, UConn Health, 263 Farmington Ave., Farmington, CT 06030-3305, USA. [19] Department of Biochemistry, University of Wisconsin-Madison, Madison, WI 53706, USA. [20] Molecular Microbiology and Structural Biochemistry, UMR5086 CNRS/Université Lyon 1, 7, passage du Vercors, 69367, Lyon, France. [21] "Rocasolano" Institute for Physical Chemistry, CSIC, 28006, Madrid, Spain. [22] Laboratory of Chemical Physics, National Institute of Diabetes and Digestive and Kidney, 20892-0520, Bethesda, USA. [23] University of Vienna, Department of Pharmaceutical Sciences, Josef-Holaubek-Platz 2, A-1090, Vienna, Austria. [24] Department of Biology, Technical University of Darmstadt, 64289, Darmstadt, Germany. [25]
DOI 10.1002/anie.202205858
PMID 36115062
发布时间 2022-12-08
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Angewandte Chemie (International ed. in English)

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