Comprehensive Fragment Screening of the SARS-CoV-2 Proteome Explores Novel Chemical Space for Drug Development.
作者:
Hannes,Berg [1]
;
Maria A,Wirtz Martin [2]
;
Nadide,Altincekic [1]
;
Islam,Alshamleh [2]
;
Jasleen,Kaur Bains [1]
;
Julius,Blechar [2]
;
Betül,Ceylan [1]
;
Vanessa,de Jesus [2]
;
Karthikeyan,Dhamotharan [1]
;
Christin,Fuks [2]
;
Santosh L,Gande [1]
;
Bruno,Hargittay [1]
;
Katharina F,Hohmann [2]
;
Marie T,Hutchison [1]
;
Sophie,Marianne Korn [2]
;
Robin,Krishnathas [2]
;
Felicitas,Kutz [3]
;
Verena,Linhard [1]
;
Tobias,Matzel [1]
;
Nathalie,Meiser [2]
;
Anna,Niesteruk [1]
;
Dennis J,Pyper [2]
;
Linda,Schulte [1]
;
Sven,Trucks [2]
;
Kamal,Azzaoui [1]
;
Marcel J J,Blommers [2]
;
Yojana,Gadiya [2]
;
Reagon,Karki [3]
;
Andrea,Zaliani [1]
;
Philip,Gribbon [2]
;
Marcius,da Silva Almeida [1]
;
Cristiane,Dinis Anobom [2]
;
Anna L,Bula [1]
;
Matthias,Bütikofer [2]
;
Ícaro,Putinhon Caruso [1]
;
Isabella,Caterina Felli [2]
;
Andrea T,Da Poian [1]
;
Gisele,Cardoso de Amorim [1]
;
Nikolaos K,Fourkiotis [2]
;
Angelo,Gallo [1]
;
Dhiman,Ghosh [2]
;
Francisco,Gomes-Neto [1]
;
Oksana,Gorbatyuk [2]
;
Bing,Hao [1]
;
Vilius,Kurauskas [4]
;
Lauriane,Lecoq [4]
;
Yunfeng,Li [5]
;
Nathane,Cunha Mebus-Antunes [6]
;
Miguel,Mompeán [5]
;
Thais,Cristtina Neves-Martins [6]
;
Martí,Ninot-Pedrosa [5]
;
Anderson S,Pinheiro [6]
;
Letizia,Pontoriero [5]
;
Yulia,Pustovalova [6]
;
Roland,Riek [7]
;
Angus J,Robertson [6]
;
Marie,Jose Abi Saad [8]
;
Miguel Á,Treviño [9]
;
Aikaterini C,Tsika [10]
;
Fabio C L,Almeida [11]
;
Ad,Bax [7]
;
Katherine,Henzler-Wildman [12]
;
Jeffrey C,Hoch [13]
;
Kristaps,Jaudzems [14]
;
Douglas V,Laurents [7]
;
Julien,Orts [7]
;
Roberta,Pierattelli [15]
;
Georgios A,Spyroulias [16]
;
Elke,Duchardt-Ferner [16]
;
Jan,Ferner [17]
;
Boris,Fürtig [11]
;
Martin,Hengesbach [8]
;
Frank,Löhr [18]
;
Nusrat,Qureshi [19]
;
Christian,Richter [19]
;
Krishna,Saxena [20]
;
Andreas,Schlundt [21]
;
Sridhar,Sreeramulu [19]
;
Anna,Wacker [7]
;
Julia E,Weigand [22]
;
Julia,Wirmer-Bartoschek [7]
;
Jens,Wöhnert [21]
;
Harald,Schwalbe [9]
作者单位:
Institute for Organic Chemistry and Chemical Biology, Goethe University Frankfurt, 60438, Frankfurt am Main, Germany.
[1]
Center of Biomolecular Magnetic Resonance (BMRZ), Goethe University Frankfurt, Frankfurt am Main (Germany), Max-von-LaueStrasse 7+9, 60438, Frankfurt am Main, Germany.
[2]
Institute for Molecular Biosciences, Goethe University Frankfurt, Max-von-Laue Strasse 7+9, 60438, Frankfurt am Main, Germany.
[3]
Saverna Therapeutics, Pumpmattenweg 3, 4105, Biel-Benken, Switzerland.
[4]
Fraunhofer Institute for Translational Medicine and Pharmacology (ITMP), Screening Port, Schnackenburgallee 114, 22525, Hamburg, Germany.
[5]
Fraunhofer Cluster of Excellence for Immune-Mediated Diseases (CIMD), Theodor-Stern-Kai 7, 60596, Frankfurt am Main, Germany.
[6]
Institute of Medical Biochemistry, Federal University of Rio de Janeiro, 21941-902, Rio de Janeiro, Brazil.
[7]
National Center of Nuclear Magnetic Resonance (CNRMN), CENABIO, Federal University of Rio de Janeiro, 21941-902, Rio de Janeiro, Brazil.
[8]
Department of Biochemistry, Institute of Chemistry, Federal University of Rio de Janeiro, 21941-902, Rio de Janeiro, Brazil.
[9]
Latvian Institute of Organic Synthesis, Aizkraukles 21, LV-1006, Riga, Latvia.
[10]
ETH, Swiss Federal Institute of Technology, Laboratory of Physical Chemistry, HCI F217, Vladimir-Prelog-Weg 2, 8093, Zürich, Switzerland.
[11]
Multiuser Center for Biomolecular Innovation (CMIB), Department of Physics, São Paulo State University (UNESP), 01049-010, São José do Rio Preto, Brazil.
[12]
Magnetic Resonance Center (CERM), University of Florence, Via Luigi Sacconi 6, Sesto Fiorentino, 50019, Florence, Italy.
[13]
Department of Chemistry "Ugo Schiff", University of Florence, Via della Lastruccia 3-13, Sesto Fiorentino, 50019, Florence, Italy.
[14]
Multidisciplinary Center for Research in Biology (NUMPEX), Campus Duque de Caxias Federal University of Rio de Janeiro, 25.250-470, Duque de Caxias, Brazil.
[15]
Department of Pharmacy, University of Patras, 26504, Patras, Greece.
[16]
Department of Chemistry, University of Torino, IT-10126, Torino, Italy.
[17]
Laboratory of Toxinology, Oswaldo Cruz Foundation (FIOCRUZ), 21040-900, Rio de Janeiro, Brazil.
[18]
Department of Molecular Biology and Biophysics, UConn Health, 263 Farmington Ave., Farmington, CT 06030-3305, USA.
[19]
Department of Biochemistry, University of Wisconsin-Madison, Madison, WI 53706, USA.
[20]
Molecular Microbiology and Structural Biochemistry, UMR5086 CNRS/Université Lyon 1, 7, passage du Vercors, 69367, Lyon, France.
[21]
"Rocasolano" Institute for Physical Chemistry, CSIC, 28006, Madrid, Spain.
[22]
Laboratory of Chemical Physics, National Institute of Diabetes and Digestive and Kidney, 20892-0520, Bethesda, USA.
[23]
University of Vienna, Department of Pharmaceutical Sciences, Josef-Holaubek-Platz 2, A-1090, Vienna, Austria.
[24]
Department of Biology, Technical University of Darmstadt, 64289, Darmstadt, Germany.
[25]
DOI
10.1002/anie.202205858
PMID
36115062
发布时间
2022-12-08
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Angewandte Chemie (International ed. in English)
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