Identification of 1,4-Benzodiazepine-2,5-dione Derivatives as Potential Protein Synthesis Inhibitors with Highly Potent Anticancer Activity.
第一作者:
Wenjun,Yu
第一单位:
School of Pharmaceutical Sciences, Tsinghua University, Haidian Dist, Beijing 100084, P. R. China.
作者:
主题词
人类(Humans);小鼠(Mice);动物(Animals);药物筛选试验, 抗肿瘤(Drug Screening Assays, Antitumor);蛋白质合成抑制药(Protein Synthesis Inhibitors);细胞增殖(Cell Proliferation);抗肿瘤药(Antineoplastic Agents);癌, 非小细胞肺(Carcinoma, Non-Small-Cell Lung);肺肿瘤(Lung Neoplasms);细胞系, 肿瘤(Cell Line, Tumor);细胞凋亡(Apoptosis);构效关系(Structure-Activity Relationship);剂量效应关系, 药物(Dose-Response Relationship, Drug);分子结构(Molecular Structure)
DOI
10.1021/acs.jmedchem.2c01431
PMID
36260776
发布时间
2022-12-04
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Journal of medicinal chemistry
14891-14915页
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