作者:
Youwen,Zhuang [1]
;
Yue,Wang [2]
;
Bingqing,He [3]
;
Xinheng,He [2]
;
X Edward,Zhou [4]
;
Shimeng,Guo [5]
;
Qidi,Rao [6]
;
Jiaqi,Yang [7]
;
Jinyu,Liu [8]
;
Qingtong,Zhou [9]
;
Xiaoxi,Wang [7]
;
Mingliang,Liu [7]
;
Weiyi,Liu [2]
;
Xiangrui,Jiang [2]
;
Dehua,Yang [10]
;
Hualiang,Jiang [11]
;
Jingshan,Shen [2]
;
Karsten,Melcher [4]
;
Hong,Chen [12]
;
Yi,Jiang [2]
;
Xi,Cheng [2]
;
Ming-Wei,Wang [13]
;
Xin,Xie [14]
;
H Eric,Xu [15]
作者单位:
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China. Electronic address: zhuangyouwen@simm.ac.cn.
[1]
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; University of Chinese Academy of Sciences, Beijing 100049, China.
[2]
University of Chinese Academy of Sciences, Beijing 100049, China; The State Key Laboratory of Drug Research, The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China.
[3]
Department of Structural Biology, Van Andel Research Institute, Grand Rapids, MI 49503, USA.
[4]
University of Chinese Academy of Sciences, Beijing 100049, China; The State Key Laboratory of Drug Research, The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing 210046, China.
[5]
School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China.
[6]
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.
[7]
School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing 210046, China.
[8]
Department of Pharmacology, School of Basic Medical Sciences, Fudan University, Shanghai 200032, China.
[9]
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; University of Chinese Academy of Sciences, Beijing 100049, China; The State Key Laboratory of Drug Research, The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.
[10]
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; University of Chinese Academy of Sciences, Beijing 100049, China; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China.
[11]
Shanghai Key Laboratory of Crime Scene Evidence, Shanghai Research Institute of Criminal Science and Technology, Shanghai 200083, China; Shanghai Yuansi Standard Science and Technology Co., Ltd, Shanghai 200080, China.
[12]
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; University of Chinese Academy of Sciences, Beijing 100049, China; The State Key Laboratory of Drug Research, The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China; Department of Pharmacology, School of Basic Medical Sciences, Fudan University, Shanghai 200032, China. Electronic address: mwwang@simm.ac.cn.
[13]
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; University of Chinese Academy of Sciences, Beijing 100049, China; The State Key Laboratory of Drug Research, The National Center for Drug Screening, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing 210046, China; School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, UCAS, Hangzhou 310024, China. Electronic address: xxie@simm.ac.cn.
[14]
The CAS Key Laboratory of Receptor Research, Center for Structure and Function of Drug Targets, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China; University of Chinese Academy of Sciences, Beijing 100049, China. Electronic address: eric.xu@simm.ac.cn.
[15]
主题词
人类(Humans);镇痛药, 阿片类(Analgesics, Opioid);抑制蛋白(Arrestin);芬太尼(Fentanyl);GTP结合蛋白质类(GTP-Binding Proteins);吗啡(Morphine);受体, 阿片样, μ(Receptors, Opioid, mu)
DOI
10.1016/j.cell.2022.09.041
PMID
36368306
发布时间
2023-01-25
- 浏览3

Cell
Cell
4361-4375.e19页
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