VIP152 is a selective CDK9 inhibitor with pre-clinical in vitro and in vivo efficacy in chronic lymphocytic leukemia.
第一作者:
Steven,Sher
第一单位:
Division of Hematology, Department of Internal Medicine, The Ohio State University College of Medicine, Columbus, OH, USA.
作者:
主题词
动物(Animals);小鼠(Mice);阳性转录延伸因子B(Positive Transcriptional Elongation Factor B);白血病, 淋巴细胞, 慢性, B细胞(Leukemia, Lymphocytic, Chronic, B-Cell);细胞周期蛋白依赖激酶9(Cyclin-Dependent Kinase 9);细胞周期蛋白T(Cyclin T);磷酰化(Phosphorylation);细胞核(Cell Nucleus);蛋白激酶抑制剂(Protein Kinase Inhibitors)
DOI
10.1038/s41375-022-01758-z
PMID
36376377
发布时间
2023-09-30
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Leukemia
326-338页
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