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Porcupine inhibitor CGX1321 alleviates heart failure with preserved ejection fraction in mice by blocking WNT signaling.

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作者单位: Department of Cardiology, Daping Hospital, Third Military Medical University (Army Military Medical University), Chongqing, 400042, China. [1] Chongqing Key Laboratory for Hypertension Research, Chongqing Cardiovascular Clinical Research Center, Chongqing Institute of Cardiology, Chongqing, 400042, China. [2] Department of Cardiovascular Medicine, The General Hospital of Western Theater Command PLA, Chengdu, 610083, China. [3] School of Medicine, Chongqing University, Chongqing, 400044, China. [4] Guangzhou Curegenix Co. Ltd., International Business Incubator, Guangzhou Science City, Guangzhou, 510663, China. [5] Curegenix, Inc., Burlingame, CA, 94010, USA. [6] Department of Cardiology, Daping Hospital, Third Military Medical University (Army Military Medical University), Chongqing, 400042, China. chunyuzeng01@163.com. [7] Chongqing Key Laboratory for Hypertension Research, Chongqing Cardiovascular Clinical Research Center, Chongqing Institute of Cardiology, Chongqing, 400042, China. chunyuzeng01@163.com. [8] State Key Laboratory of Trauma, Burns and Combined Injury, Daping Hospital, The Third Military Medical University, Chongqing, 400042, China. chunyuzeng01@163.com. [9] Heart Center of Fujian Province, Union Hospital, Fujian Medical University, Fuzhou, 350001, China. chunyuzeng01@163.com. [10] Department of Cardiology, Chongqing General Hospital, Chongqing, 401147, China. chunyuzeng01@163.com. [11] Cardiovascular Research Center of Chongqing College, Chinese Academy of Sciences, University of Chinese Academy of Sciences, Chongqing, 400722, China. chunyuzeng01@163.com. [12] Department of Cardiology, Daping Hospital, Third Military Medical University (Army Military Medical University), Chongqing, 400042, China. weiericwang@163.com. [13] Chongqing Key Laboratory for Hypertension Research, Chongqing Cardiovascular Clinical Research Center, Chongqing Institute of Cardiology, Chongqing, 400042, China. weiericwang@163.com. [14] Department of Geriatrics, Southwest Hospital, Third Military Medical University (Army Medical University), Chongqing, 400038, China. weiericwang@163.com. [15]
DOI 10.1038/s41401-022-01025-y
PMID 36473990
发布时间 2024-06-03
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Acta pharmacologica Sinica

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