Design, Synthesis, Molecular Docking, and Biological Evaluation of Novel Pimavanserin-Based Analogues as Potential Serotonin 5-HT<sub>2A</sub> Receptor Inverse Agonists.
作者:
主题词
人类(Humans);血清素(Serotonin);药物反向激动作用(Drug Inverse Agonism);受体, 血清素, 5-HT2A(Receptor, Serotonin, 5-HT2A);血清素5-HT2受体激动剂(Serotonin 5-HT2 Receptor Agonists);精神病(Psychotic Disorders);血清素受体激动剂(Serotonin Receptor Agonists);尿素(Urea);抗精神病药(Antipsychotic Agents)
DOI
10.1021/acs.jmedchem.3c00662
PMID
37378639
发布时间
2023-07-18
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Journal of medicinal chemistry
9057-9075页
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