作者:
Simone,Bonazzi [1]
;
Audrey,Gray [2]
;
Noel M,Thomsen [1]
;
Jonathan,Biag [2]
;
Nancy,Labbe-Giguere [1]
;
Erin P,Keaney [1]
;
Hasnain A,Malik [1]
;
Yingchuan,Sun [1]
;
Jill,Nunez [1]
;
Rajeshri G,Karki [1]
;
Mark,Knapp [3]
;
Robert,Elling [3]
;
John,Fuller [4]
;
Gwynn,Pardee [4]
;
Lucas,Craig [2]
;
Ketthsy,Capre [2]
;
Sarah,Salas [2]
;
Aakruti,Gorde [2]
;
Guiqing,Liang [5]
;
Danuta,Lubicka [6]
;
Stephanie M,McTighe [2]
;
Carleton,Goold [2]
;
Shanming,Liu [7]
;
Lin,Deng [5]
;
Jin,Hong [8]
;
Alexander,Fekete [8]
;
Pascal,Stadelmann [9]
;
Wilfried,Frieauff [9]
;
Azeddine,Elhajouji [9]
;
Daniel,Bauer [9]
;
Andreas,Lerchner [10]
;
Branko,Radetich [1]
;
Pascal,Furet [10]
;
Grazia,Piizzi [1]
;
Doug,Burdette [5]
;
Christopher J,Wilson [2]
;
Stefan,Peukert [1]
;
Lawrence G,Hamann [1]
;
Leon O,Murphy [7]
;
Daniel,Curtis [2]
作者单位:
Global Discovery Chemistry, Novartis Institutes for BioMedical Research, 181 Massachusetts Ave, Cambridge, Massachusetts 02139, United States.
[1]
Neuroscience, Novartis Institutes for BioMedical Research, 22 Windsor Street, Cambridge, Massachusetts 02139, United States.
[2]
Global Discovery Chemistry, Novartis Institutes for BioMedical Research, 5959 Horton St, Emeryville, California 94608, United States.
[3]
Chemical Biology and Therapeutics, Novartis Institutes for BioMedical Research, 5959 Horton St, Emeryville, California 94608, United States.
[4]
Pharmacokinetic Sciences, Novartis Institutes for BioMedical Research, 250 Massachusetts Avenue, Cambridge, Massachusetts 02139, United States.
[5]
Global Drug Development/Technical Research and Development, Novartis Institutes for BioMedical Research, 700 Main Street, Cambridge, Massachusetts 02139, United States.
[6]
Chemical Biology and Therapeutics, Novartis Institutes for BioMedical Research, 181 Massachusetts Ave, Cambridge, Massachusetts 02139, United States.
[7]
Preclinical Safety, Novartis Institutes for BioMedical Research, 250 Massachusetts Avenue, Cambridge, Massachusetts 02139, United States.
[8]
Preclinical Safety, Novartis Institutes for BioMedical Research, Fabrikstrasse 28, 4056 Basel, Switzerland.
[9]
Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Fabrikstrasse 22, 4056 Basel, Switzerland.
[10]
主题词
小鼠(Mice);动物(Animals);西罗莫司(Sirolimus);综合征(Syndrome);中枢神经系统(Central Nervous System);脑(Brain);TOR丝氨酸-苏氨酸激酶(TOR Serine-Threonine Kinases);腺苷三磷酸(Adenosine Triphosphate)
DOI
10.1021/acs.jmedchem.3c00705
PMID
37399505
发布时间
2023-07-18
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Journal of medicinal chemistry
Journal of medicinal chemistry
9095-9119页
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